Pay in 4 interest-free payments of $25.00 Learn more
Ships within 48 hours · Estimated delivery Aug 2 - Aug 7
Formula: C16H8Br2F6N6O
InChiKey: ALIVXCSEERJYHU-UHFFFAOYSA-N
Chemical Name: N-{17
Smiles: C[C@@]12O[C@H]1[C@H](C)[C@@H]1C[C@@](O)(NC(=O)O1)[C@@H](C=CC=C(C)CC1C=C(C(Cl)=C(C=1)OC)N(C)C(=O)C[C@@H]2OC(=O)[C@H](C)N(C)C(=O)CCCCCN1C(=O)C=CC1=O)OC |c:17
PCS1055 dihydrochloride Catalog No.:M32998-C Formula: C16H8Br2F6N6OPCS1055 dihydrochloride is a potent, selective and competitive muscarinic M4 receptor antagonist with an IC50 of 18. 1 nM and a Kd of 5. 72 nM. PCS1055 dihydrochloride inhibits radioligand [3H] NMS binding to the M4 receptor with a Ki of 6. 5 nM. PCS1055 dihydrochloride exhibits >100 fold selectivity over M1 , M3 , and M5 receptors and 30 fold selectivity at the M2 receptor. PCS1055 dihydrochloride is also a potent AChE inhibitor with IC50 s of 22 nM